The davis-beirut reaction: A novel entry into 2h-indazoles and indazolones. Recent biological activity of indazoles

Makhluf J. Haddadin, Wayne E. Conrad, Mark J. Kurth

Research output: Contribution to journalArticle

47 Citations (Scopus)

Abstract

A novel, easy method for the syntheses of richly diversified 2H-indazoles and indazolones, called the Davis-Beirut reaction, and other recent 2H-indazole synthetic routes are briefly reviewed. An update on the biological activity of indazoles is also surveyed.

Original languageEnglish (US)
Pages (from-to)1293-1300
Number of pages8
JournalMini-Reviews in Medicinal Chemistry
Volume12
Issue number12
DOIs
StatePublished - 2012

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Indazoles

Keywords

  • 2H-indazoles
  • Biological activity
  • Davis-beirut reaction
  • Indazolone

ASJC Scopus subject areas

  • Pharmacology
  • Drug Discovery

Cite this

The davis-beirut reaction : A novel entry into 2h-indazoles and indazolones. Recent biological activity of indazoles. / Haddadin, Makhluf J.; Conrad, Wayne E.; Kurth, Mark J.

In: Mini-Reviews in Medicinal Chemistry, Vol. 12, No. 12, 2012, p. 1293-1300.

Research output: Contribution to journalArticle

Haddadin, Makhluf J. ; Conrad, Wayne E. ; Kurth, Mark J. / The davis-beirut reaction : A novel entry into 2h-indazoles and indazolones. Recent biological activity of indazoles. In: Mini-Reviews in Medicinal Chemistry. 2012 ; Vol. 12, No. 12. pp. 1293-1300.
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