Abstract
A one-step heterocyclization of o-nitrobenzylamines to 3-alkoxy-2H- indazoles is reported. The electronic nature of the nitrophenyl group, the steric and electronic nature of the R1-functionalized benzylic amine, and the nature of the alcoholic solvent affect the efficiency of this heterocyclization reaction (∼40-90%).
Original language | English (US) |
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Pages (from-to) | 2687-2689 |
Number of pages | 3 |
Journal | Journal of Organic Chemistry |
Volume | 71 |
Issue number | 7 |
DOIs | |
State | Published - Apr 1 2006 |
ASJC Scopus subject areas
- Organic Chemistry