Inverse electron demand diels-alder reactions of indole IV. A new route to β-carbolines

Wen Hong Fan; Mamta Parikh; John K. Snyder

doi:10.1016/00404-0399(50)1347-K

Inverse electron demand diels-alder reactions of indole IV. A new route to β-carbolines

Wen Hong Fan, Mamta Parikh, John K. Snyder

Research output: Contribution to journal › Article

25 Scopus citations

Abstract

β-Carbolines have been prepared by the intramolecular cycloaddition of indole with 1,2,4-triazines tethered from C3 with the indolyl nitrogen using a thiourea linkage. Subsequent to the cycloaddition, reductive cleavage of the thiourea subunit provides the βcarboline.

Original language	English (US)
Pages (from-to)	6591-6594
Number of pages	4
Journal	Tetrahedron Letters
Volume	36
Issue number	37
DOIs	https://doi.org/10.1016/00404-0399(50)1347-K
State	Published - Jan 1 1995
Externally published	Yes

Fingerprint

ASJC Scopus subject areas

Biochemistry
Drug Discovery
Organic Chemistry

Cite this

Fan, W. H., Parikh, M., & Snyder, J. K. (1995). Inverse electron demand diels-alder reactions of indole IV. A new route to β-carbolines. Tetrahedron Letters, 36(37), 6591-6594. https://doi.org/10.1016/00404-0399(50)1347-K

@article{ce35b62b4d3f44f78934b2d643cd8113,

title = "Inverse electron demand diels-alder reactions of indole IV. A new route to β-carbolines",

abstract = "β-Carbolines have been prepared by the intramolecular cycloaddition of indole with 1,2,4-triazines tethered from C3 with the indolyl nitrogen using a thiourea linkage. Subsequent to the cycloaddition, reductive cleavage of the thiourea subunit provides the βcarboline.",

author = "Fan, {Wen Hong} and Mamta Parikh and Snyder, {John K.}",

year = "1995",

month = jan

day = "1",

doi = "10.1016/00404-0399(50)1347-K",

language = "English (US)",

volume = "36",

pages = "6591--6594",

journal = "Tetrahedron Letters",

issn = "0040-4039",

publisher = "Elsevier Limited",

number = "37",

}

TY - JOUR

T1 - Inverse electron demand diels-alder reactions of indole IV. A new route to β-carbolines

AU - Fan, Wen Hong

AU - Parikh, Mamta

AU - Snyder, John K.

PY - 1995/1/1

Y1 - 1995/1/1

N2 - β-Carbolines have been prepared by the intramolecular cycloaddition of indole with 1,2,4-triazines tethered from C3 with the indolyl nitrogen using a thiourea linkage. Subsequent to the cycloaddition, reductive cleavage of the thiourea subunit provides the βcarboline.

AB - β-Carbolines have been prepared by the intramolecular cycloaddition of indole with 1,2,4-triazines tethered from C3 with the indolyl nitrogen using a thiourea linkage. Subsequent to the cycloaddition, reductive cleavage of the thiourea subunit provides the βcarboline.

UR - http://www.scopus.com/inward/record.url?scp=0029143822&partnerID=8YFLogxK

UR - http://www.scopus.com/inward/citedby.url?scp=0029143822&partnerID=8YFLogxK

U2 - 10.1016/00404-0399(50)1347-K

DO - 10.1016/00404-0399(50)1347-K

M3 - Article

AN - SCOPUS:0029143822

VL - 36

SP - 6591

EP - 6594

JO - Tetrahedron Letters

JF - Tetrahedron Letters

SN - 0040-4039

IS - 37

ER -

Access to Document

10.1016/00404-0399(50)1347-K