Abstract
β-Carbolines have been prepared by the intramolecular cycloaddition of indole with 1,2,4-triazines tethered from C3 with the indolyl nitrogen using a thiourea linkage. Subsequent to the cycloaddition, reductive cleavage of the thiourea subunit provides the βcarboline.
| Original language | English (US) |
|---|---|
| Pages (from-to) | 6591-6594 |
| Number of pages | 4 |
| Journal | Tetrahedron Letters |
| Volume | 36 |
| Issue number | 37 |
| DOIs | |
| State | Published - Jan 1 1995 |
| Externally published | Yes |
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ASJC Scopus subject areas
- Biochemistry
- Drug Discovery
- Organic Chemistry
Cite this
Inverse electron demand diels-alder reactions of indole IV. A new route to β-carbolines. / Fan, Wen Hong; Parikh, Mamta; Snyder, John K.
In: Tetrahedron Letters, Vol. 36, No. 37, 01.01.1995, p. 6591-6594.Research output: Contribution to journal › Article
}
TY - JOUR
T1 - Inverse electron demand diels-alder reactions of indole IV. A new route to β-carbolines
AU - Fan, Wen Hong
AU - Parikh, Mamta
AU - Snyder, John K.
PY - 1995/1/1
Y1 - 1995/1/1
N2 - β-Carbolines have been prepared by the intramolecular cycloaddition of indole with 1,2,4-triazines tethered from C3 with the indolyl nitrogen using a thiourea linkage. Subsequent to the cycloaddition, reductive cleavage of the thiourea subunit provides the βcarboline.
AB - β-Carbolines have been prepared by the intramolecular cycloaddition of indole with 1,2,4-triazines tethered from C3 with the indolyl nitrogen using a thiourea linkage. Subsequent to the cycloaddition, reductive cleavage of the thiourea subunit provides the βcarboline.
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UR - http://www.scopus.com/inward/citedby.url?scp=0029143822&partnerID=8YFLogxK
U2 - 10.1016/00404-0399(50)1347-K
DO - 10.1016/00404-0399(50)1347-K
M3 - Article
VL - 36
SP - 6591
EP - 6594
JO - Tetrahedron Letters
JF - Tetrahedron Letters
SN - 0040-4039
IS - 37
ER -